Current landscape of phosphodiesterase 10A (PDE10A) inhibition

J Med Chem. 2012 Sep 13;55(17):7299-331. doi: 10.1021/jm3004976. Epub 2012 Aug 14.
No abstract available

MeSH terms

  • Animals
  • Cyclic AMP / metabolism
  • Cyclic GMP / metabolism
  • Humans
  • Hydrolysis
  • Mice
  • Models, Molecular
  • Phosphodiesterase Inhibitors / pharmacology*
  • Phosphoric Diester Hydrolases / chemistry
  • Phosphoric Diester Hydrolases / drug effects*
  • Rats

Substances

  • Phosphodiesterase Inhibitors
  • Cyclic AMP
  • PDE10A protein, human
  • Phosphoric Diester Hydrolases
  • Cyclic GMP