Agents used in N2a-based pharmacological screens.
Agent | Primary Target | Other targets | Suppliers |
---|---|---|---|
Rapamycin | mTORC1 | mTORC2 | A.G. Scientific, R-1018 |
Bisindolylmaleimide V (B5) | S6K1 | Unknown | Enzo Life, ALX-270-053 Sciences |
CX-4945 | CK2 | DYRK2 | Selleckchem, S2248 |
TBB | CK2 | DYRK2, PIM | Tocris, 2275 |
DRB | CDK7/CK2 | CDK8, CDK9 | EMD Millipore, 287891 |
PHA-767491 | Cdc7 | CDK9, MK2 | Tocris, 3140 |
D4476 | CK1 | ALK5, PKD1, p38a | Tocris, 2902 |
IC261 | CK1 | PKA. Fyn | EMD Millipore, 400090 |
Staurosporine | Pan Kinase | PP1 | Tocris, 1285 |