Table 2

Summary of agonist-antagonist interactions on EUS function.

DrugsEUS
AgonistAntagonistBurstingTonic Activity
L-DOPA
(DA precursor)
Increased (+)Suppressed (–)
SCH 23390
(DR1 antagonist)
ReversesReverses
Remoxipride
(DR2 antagonist)
No effectSlightly increased
APO
(DR antagonist)
Increased (+)Suppressed (–)
SCH 23390
(DR1 antagonist)
ReversesReverses
Remoxipride
(DR2 antagonist)
No effectSlightly increased
Quinpirole
(DR2 agonist)
Increased (+)No effect
Remoxipride
(DR2 antagonist)
ReversesNo effect